Peptide Profile

TB-500

A powerful fragment of thymosin beta-4 that acts like your body's repair signal—speeding up healing of muscles, tendons, and tissues by promoting cell migration and new blood vessel growth right where you need it most.

Healing & Recovery

Dose Range

2-5mg

Frequency

Twice weekly

Route

Subcutaneous injection

Cycle Length

4-6 weeks

Onset

Moderate (1-2 weeks)

Evidence

Moderate

Compound Profile

Scientific & Efficacy Data

C38H68N10O14

Molecular Formula

889.01 g/mol

Molecular Weight

2-3 days (systemic)

Half-Life

High via subcutaneous injection (~100%)

Bioavailability

885340-08-9

CAS #

66356057

PubChem ID ↗

Developed By · 1981

Allan L. Goldstein, PhD

George Washington University School of Medicine

Primary Benefits

Healing Speed

Accelerates tissue repair through cell migration and angiogenesis—one of the most effective peptides for injury recovery

Tissue Repair

Regenerates muscle, tendon, and ligament tissue by promoting new blood vessel formation and reducing inflammation

Anti-Scarring

Prevents fibroblast-to-myofibroblast conversion, reducing scar tissue formation and preserving tissue flexibility

Amino Acid Sequence

Ac-LKKTETQ (N-Acetyl-Leu-Lys-Lys-Thr-Glu-Thr-Gln)

Dosing

How much
do I take?

Starting Dose

2-2.5 mg

Frequency

Twice weekly

Duration

4-6 weeks

Start here to assess your tolerance and response. Many people see good results at this dose. Split your weekly dose into two injections spaced 3-4 days apart (like Monday and Thursday).

Standard Dose

4-5 mg

Frequency

Twice weekly (split into 2-2.5 mg doses)

Duration

4-6 weeks

The most commonly used protocol for moderate injuries. Your total weekly dose is 4-5 mg, split into two injections. This is the sweet spot where most users see significant healing benefits.

Advanced Dose

5-10 mg

Frequency

Twice weekly (2.5-5 mg per injection)

Duration

4-8 weeks

Higher doses for severe or stubborn injuries. Some protocols use a loading phase of higher doses for 1-2 weeks, then drop to maintenance. Work with a provider for doses above 5 mg weekly.

Timing

Best time to take

Morning or evening—timing doesn't significantly affect TB-500's effectiveness. What matters most is consistency. Pick a schedule that works for your lifestyle and stick with it.

With food?

TB-500 can be injected regardless of food timing. It doesn't seem to affect absorption either way, so fit it into whatever routine works for you.

If stacking

TB-500 pairs exceptionally well with BPC-157—they're often called the 'healing stack' because they work through different but complementary mechanisms. Inject at different sites if using both. Space injections at least 15-30 minutes apart to track individual effects.

Adjusting Your Dose

Increase if

  • +You've completed 2+ weeks at starting dose with minimal healing progress
  • +Your injury is more severe than initially assessed
  • +You're recovering from surgery under professional guidance
  • +Your research protocol calls for loading phases

Decrease if

  • -You experience persistent headaches or fatigue beyond the first week
  • -Injection site reactions don't resolve within 48 hours
  • -You feel unusually tired or lethargic after each injection
  • -Any unexpected or uncomfortable side effects arise

Signs of right dose

  • Noticeable improvement in injury flexibility or reduced stiffness
  • Decreased pain at the injury site over 2-4 weeks
  • Improved range of motion in affected areas
  • Better exercise tolerance without aggravating the injury

Dosing Calculator

Calculate Your Exact Dose

Peptide in Vial

mg

BAC Water Added

2ml
ml

Desired Dose

mcg

Amount to Draw

10

units

0.0ml0.1ml0.2ml0.3ml0.4ml0.5ml0.6ml0.7ml0.8ml0.9ml1.0ml
0102030405060708090100

Concentration

2.50 mg/ml (2500 mcg/ml)

Suitability

Is this
right for me?

Best For

Athletes Recovering from Muscle Injuries

If you've pulled a hamstring, strained your back, or torn a muscle, TB-500 helps accelerate the healing process by promoting cell migration to the injury site and supporting new blood vessel growth. It's especially useful for injuries that just won't seem to fully heal.

Tendon and Ligament Problems

Tendons and ligaments are notoriously slow healers because they have poor blood supply. TB-500 promotes angiogenesis (new blood vessel formation) and helps repair these stubborn connective tissue injuries—think Achilles tendonitis, tennis elbow, or rotator cuff issues.

Post-Surgical Recovery

After surgery, your body needs to repair a lot of tissue quickly. TB-500 supports wound healing, reduces inflammation, and may help minimize scar tissue formation. Some protocols use it alongside traditional recovery to potentially speed up the healing timeline.

Chronic Inflammation and Slow Healers

Some people just heal slowly—whether due to age, diabetes, or other factors. TB-500 helps regulate the inflammatory response and promotes the cellular processes needed for tissue repair. It essentially tells your body to focus healing resources where they're needed most.

Consider Alternatives If

Goal: General tissue healing and gut support

Consider: BPC-157, Pentadecapeptide, GHK-Cu

Goal: Muscle recovery and growth

Consider: IGF-1 LR3, MGF (Mechano Growth Factor), GHRP peptides

Goal: Wound healing and skin repair

Consider: GHK-Cu, BPC-157, Collagen peptides

Who Should Avoid

Do not use if

  • ×You are pregnant or might become pregnant—we don't know how TB-500 affects fetal development
  • ×You are breastfeeding—the peptide could potentially pass into breast milk
  • ×You have active cancer or a history of cancer—angiogenesis promotion is concerning in cancer contexts
  • ×You've ever had a serious allergic reaction to any peptide
  • ×You're under 18—TB-500 is for adult use only in research settings
  • ×You have an active infection at the injury site—heal the infection first

Use with caution if

  • !You take blood thinners like warfarin or aspirin—may increase bleeding at injection sites
  • !You have cardiovascular conditions—discuss with your doctor first
  • !You're diabetic—some peptides can affect healing and blood sugar
  • !You have autoimmune conditions—immune modulation effects may be unpredictable
  • !You're taking NSAIDs regularly—these may interfere with the healing cascade
  • !You have a history of blood clots—angiogenesis effects need consideration

Not Sure?

Compare TB-500 with similar peptides to find the best fit for your goals.

Administration

How do I
use it?

Reconstitution

What you need

  • Bacteriostatic water (BAC water)—the preservative keeps it safe for multiple uses
  • Insulin syringes (29-31 gauge)—thin needles mean less discomfort
  • Alcohol swabs for cleaning vial tops and injection sites
  • Your TB-500 powder vial

Example

If you have a 5mg vial and add 2mL of BAC water, you get a concentration of 2.5mg/mL. So every 1mL (100 units on an insulin syringe) equals 2.5mg of TB-500.

For a 2.5mg dose at 2.5mg/mL concentration: draw 1mL (100 units on a standard insulin syringe). For a 5mg dose: draw the full 2mL or use a larger vial reconstituted accordingly.

Injection

Route

Subcutaneous injection (just under the skin)—the easiest and most common method. Some users prefer injecting near the injury site, though systemic administration works well too.

Best sites

  • Belly fat area (about 2 inches away from your belly button)
  • Front or outer thigh (middle section)
  • Near the injury site (within a few inches, not directly into it)
  • Back of the upper arm (have someone help if needed)

Technique

  • 1.Wash your hands thoroughly with soap and water
  • 2.Clean the injection site with an alcohol swab and let it air dry completely
  • 3.Pinch about an inch of skin to create a fold
  • 4.Insert the needle at a 45-90 degree angle (45 if you're lean, 90 if you have more tissue)
  • 5.Push the plunger slowly and steadily
  • 6.Wait 5 seconds before removing the needle
  • 7.Apply light pressure if needed—don't rub

Storage

Before reconstitution

Keep your TB-500 powder in the refrigerator (36-46°F / 2-8°C) for short-term storage or in the freezer (-4°F / -20°C) for long-term storage. Store in the original sealed vial away from light. Properly stored powder can remain stable for 2+ years when frozen.

After reconstitution

Once mixed with bacteriostatic water, refrigerate at 36-46°F (2-8°C). Never freeze the reconstituted solution—freezing destroys the peptide. Keep away from light and use within 28 days.

Signs of degradation

  • Cloudy or hazy appearance (should be crystal clear)
  • Visible particles floating or settled at the bottom
  • Color changes—any yellowing or discoloration means toss it
  • Unusual smell—fresh solution should have little to no odor

Sample Daily Schedule

Morning (or consistent time that works for you)

2-2.5 mg injection

Site: Rotate between belly, thigh, and near injury site

Inject twice weekly, spacing doses 3-4 days apart (e.g., Monday and Thursday). A typical loading phase uses 4-5 mg total per week for 4-6 weeks, followed by maintenance of 2-4 mg weekly if continued.

Safety

Is it
safe?

Safety Profile

TB-500 has shown a good safety profile across preclinical studies and limited human research. It's a fragment of thymosin beta-4, a naturally occurring protein in your body involved in healing. Most side effects are mild and transient, primarily injection site reactions. However, large-scale clinical trials are still needed to fully establish its safety profile in humans.

TB-500 has been used extensively in equine medicine and has been the subject of multiple human clinical trials for conditions like dry eye, wound healing, and cardiac repair. Phase 1-2 trials have shown it to be well-tolerated, but Phase 3 data is limited. Always work with a healthcare provider when using research compounds.

Common Side Effects

Experienced by some users

Injection site redness

A little pink or red area where you injected is totally normal. It's just your skin reacting to the needle and solution.

Management: Rotate injection sites between belly, thigh, and arm. A cool compress can help. Usually fades within 24-48 hours.

Mild fatigue or lethargy

Some users feel a bit tired after injections, especially in the first week. Your body is mobilizing healing resources.

Management: Inject in the evening if fatigue bothers you. Stay well-rested and this typically improves after the first week.

Mild headache

Occasional headaches have been reported, usually mild and in the first few days of use.

Management: Stay well-hydrated and rest if needed. These typically resolve within the first week as your body adjusts.

Slight flushing

Some users notice mild warmth or flushing at the injection site or generally, usually brief.

Management: This typically passes within 30 minutes. Not a cause for concern unless it's severe or persistent.

Less Common

  • Head rush or lightheadedness
  • Temporary nausea

These typically resolve with continued use or dose adjustment.

Stop and Seek Help If

  • ×Any signs of allergic reaction—stop immediately and seek medical help
  • ×Persistent headaches or fatigue that don't improve after the first week
  • ×Significant injection site reactions that spread or don't heal
  • ×Any side effect that feels serious or really concerns you
  • ×Your injury has healed satisfactorily
  • ×Your research protocol/cycle is complete

TB-500 is a research compound, not an FDA-approved medication. Never start, stop, or change your dosing without guidance from a qualified healthcare provider. This information is for educational purposes only—not medical advice.

Interactions

With other peptides

  • Excellent pairing—the classic 'healing stack.' BPC-157 works through different pathways and together they provide comprehensive tissue repair support. Inject at different sites.
  • Safe to combine for comprehensive tissue repair. GHK-Cu focuses on skin and collagen while TB-500 works on deeper tissue healing.
  • Can be combined for enhanced muscle recovery. Both promote tissue repair through different mechanisms.
  • Safe to stack for overall recovery. Growth hormone releasing peptides complement TB-500's healing effects.

With medications

  • !Blood thinners (warfarin, heparin) - May increase bleeding at injection sites. TB-500 promotes angiogenesis which could theoretically affect clotting. Monitor closely.
  • NSAIDs (ibuprofen, naproxen) - NSAIDs reduce inflammation which is part of the healing process TB-500 supports. May reduce effectiveness—use sparingly.
  • Corticosteroids - Steroids can impair healing. If you're on long-term steroids, discuss with your doctor.
  • Diabetes medications - TB-500 supports wound healing in diabetics but monitor blood sugar as healing processes can affect glucose.

With supplements

  • Collagen peptides - Complementary—collagen provides building blocks while TB-500 promotes the repair process.
  • Omega-3 fatty acids - Safe and potentially beneficial. Omega-3s support anti-inflammatory pathways that complement healing.
  • Vitamin C - Supports collagen synthesis and healing. Good addition to a recovery protocol.
  • Turmeric/Curcumin - Anti-inflammatory but work differently than NSAIDs. Generally considered safe to combine.

Effectiveness

Does it
work?

Evidence Level

Moderate human trials

What this means

Think of TB-500 as your body's 'come here and help' signal for healing. When you get injured, your body naturally releases thymosin beta-4 to start the repair process. TB-500 is a synthetic version of the most active part of this protein. It works by telling your cells to migrate to the injury site, promoting the growth of new blood vessels to bring oxygen and nutrients, and reducing inflammation so healing can happen properly. It also helps prevent excessive scar tissue formation, so you heal with more functional tissue instead of stiff scar tissue. It's like giving your body's repair crew a megaphone and extra supplies.

What to Expect

Week 1

What you might notice

  • Mild injection site redness (totally normal)
  • Possibly some initial fatigue or mild headache
  • Slight reduction in inflammation at injury site
  • Your body is just getting introduced to the peptide

What's normal

  • Minor injection site reactions that fade within a day
  • Feeling a bit tired on injection days
  • No dramatic changes yet—healing takes time

What's next

  • Keep following your protocol consistently
  • Track any changes in your injury or range of motion
  • Side effects typically improve after the first week

Weeks 2-3

What you might notice

  • Reduced stiffness around the injury
  • Improved flexibility or range of motion
  • Decreased pain with movement
  • Less swelling if inflammation was present

What's normal

  • Gradual improvement rather than sudden changes
  • Good days and less-good days are normal
  • Injury still present but progressing

What's next

  • Continue your protocol through the full cycle
  • Begin gentle movement or rehab exercises if appropriate
  • Don't push the injury too hard yet

Weeks 4-6

What you might notice

  • Significant improvement in injury healing
  • Better function of the affected area
  • Reduced or resolved pain
  • Ability to return to normal activities gradually

What's normal

  • Major improvement for most users by week 4-6
  • Some stubborn injuries may need extended protocols
  • Complete healing of muscle injuries, continued progress on tendons

What's next

  • Complete your cycle and assess results
  • Transition to maintenance dose if needed
  • Resume full activity cautiously with proper rehabilitation

Signs It's Working

Injury Recovery Indicators

  • Reduced pain at the injury site
  • Improved range of motion in affected joints
  • Decreased stiffness, especially in the morning
  • Less swelling and inflammation
  • Better function during daily activities

Healing Progress

  • Wounds closing more quickly than expected
  • Reduced bruising duration
  • Faster return to physical activities
  • Less need for pain medication
  • Improved tissue flexibility

Physical Performance

  • Ability to exercise without aggravating injury
  • Improved strength in previously injured area
  • Better recovery between workouts
  • Reduced compensation patterns from injury

Not Seeing Results?

Common reasons

  • Not giving it enough time—TB-500 works over weeks, not days. Tendons especially take 4-8 weeks to show major improvement
  • Dose too low for the injury severity—stubborn injuries may need higher loading doses initially
  • Poor quality peptide from unreliable source—always get third-party testing certificates (COAs)
  • Improper storage degraded the peptide—check if your solution looks clear before using
  • Still aggravating the injury with activity—healing peptides work best when you give the injury rest
  • NSAIDs blocking the healing process—these anti-inflammatory drugs can interfere with tissue repair signals

Key Research

"Thymosin beta4: a multi-functional regenerative peptide. Basic properties and clinical applications"

Goldstein AL, Hannappel E, Sosne G, 2012

Finding: This comprehensive review showed that thymosin beta-4 plays a vital role in tissue repair and regeneration. It protects cells from damage, reduces inflammation, promotes cell migration for healing, and helps form new blood vessels. The peptide also reduces scar formation by preventing fibroblasts from becoming scar-producing cells.

View Study

"Advances in the basic and clinical applications of thymosin beta4"

Goldstein AL, Kleinman HK, 2015

Finding: This update summarized decades of research showing TB4's effectiveness in directing stem cell maturation and tissue repair. Multiple clinical trials demonstrated benefits for eye injuries, skin wounds, and cardiac repair. The peptide shows potential for new applications including kidney and liver disease, spinal cord injury, and bone healing.

View Study

"Neuroprotective and neurorestorative effects of thymosin beta4 treatment following experimental traumatic brain injury"

Xiong Y, Mahmood A, Meng Y, et al., 2012

Finding: In brain injury models, thymosin beta-4 showed remarkable neuroprotective effects. It reduced cell death, decreased inflammation, promoted blood vessel formation, wound healing, and stem cell differentiation. The research provides scientific foundation for potential use in treating traumatic brain injury.

View Study

"Thymosin beta4 and the anti-fibrotic switch"

Kleinman HK, Kulik V, Goldstein AL, 2023

Finding: This study revealed TB4's powerful anti-scarring effects. It works by reducing inflammatory cell infiltration, lowering TGF-beta levels, and preventing fibroblasts from converting to myofibroblasts (scar-producing cells). The N-terminal fragment Ac-SDKP not only prevents fibrosis but can actually reverse existing scar tissue.

View Study

"Thymosin beta4 promotes endothelial progenitor cell angiogenesis via a vascular endothelial growth factor-dependent mechanism"

Zhao Y, Song J, Bi X, et al., 2018

Finding: Researchers discovered that TB4 significantly improves blood vessel formation by enhancing the function of endothelial progenitor cells. It works through the VEGF pathway, which is crucial for delivering nutrients and oxygen to healing tissues. When transplanted into damaged heart tissue, TB4-treated cells showed much better blood vessel formation.

View Study

Frequently Asked Questions

Medical Disclaimer

TB-500 is an investigational research compound not approved by the FDA for human therapeutic use. This information is for educational purposes only and should not be construed as medical advice. Always consult with a qualified healthcare provider before starting any new supplement or treatment protocol.

Last updated: 1/19/2026